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Talabostat - BioXcel Therapeutics

Drug Profile

Talabostat - BioXcel Therapeutics

Alternative Names: BXCL 701; PT-100; Talabostat mesilate; Talabostat mesylate; Val-boro-Pro

Latest Information Update: 15 Feb 2024

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At a glance

  • Originator Tufts University School of Medicine
  • Developer BioXcel Therapeutics; Georgetown University; M. D. Anderson Cancer Center; Midatech Pharma US; National Cancer Institute (USA); OnkosXcel Therapeutics
  • Class Antineoplastics; Boronic acids; Dipeptides; Pyrrolidines; Small molecules
  • Mechanism of Action Dipeptidyl peptidase 4 inhibitors; Dipeptidyl peptidase 8 inhibitors; Dipeptidyl peptidase 9 inhibitors; Fibroblast activation protein antagonists
  • Orphan Drug Status

    Orphan designation is assigned by a regulatory body to encourage companies to develop drugs for rare diseases.

    Yes - Acute myeloid leukaemia; Malignant melanoma; Pancreatic cancer; Soft tissue sarcoma
  • New Molecular Entity Yes

Highest Development Phases

  • Phase II Adenocarcinoma; Prostate cancer; Solid tumours
  • Phase I/II Pancreatic cancer
  • Phase I Acute myeloid leukaemia; Myelodysplastic syndromes
  • Preclinical Small cell lung cancer; Soft tissue sarcoma
  • Discontinued Chronic lymphocytic leukaemia; Malignant melanoma; Neutropenia; Non-small cell lung cancer

Most Recent Events

  • 12 Feb 2024 Talabostat - BioXcel Therapeutics receives Fast Track designation for Prostate cancer [PO,Tablet] (Hormone refractory, Combination therapy, Second-line therapy or greater, Treatment-naive) in USA
  • 10 Oct 2023 Efficacy data from a phase IIb trial in Prostate cancer released by BioXcel Therapeutics
  • 01 Jul 2023 Phase-II clinical trials in Adenocarcinoma (Combination therapy, Metastatic disease, Second-line therapy or greater) in USA (PO) (NCT05558982)
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