Telotristat etiprate - Lexicon Pharmaceuticals

Drug Profile

Telotristat etiprate - Lexicon Pharmaceuticals

Alternative Names: LP-778914; LX-1032; LX-1606; LX1032 hippurate; LX1606 hippurate; Telotristat ethyl; Xermelo

Latest Information Update: 09 Nov 2017

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At a glance

  • Originator Lexicon Pharmaceuticals
  • Developer Ipsen; Lexicon Pharmaceuticals
  • Class Pyrazoles; Pyrimidines; Small molecules
  • Mechanism of Action Serotonin modulators; TPH1 protein inhibitors
  • Orphan Drug Status

    Orphan designation is assigned by a regulatory body to encourage companies to develop drugs for rare diseases.

    Yes - Malignant carcinoid syndrome
  • New Molecular Entity Yes

Highest Development Phases

  • Marketed Malignant carcinoid syndrome
  • Discontinued Ulcerative colitis

Most Recent Events

  • 08 Nov 2017 Launched for Malignant carcinoid syndrome (Adjunctive treatment, Treatment-experienced) in United Kingdom, Germany (PO)
  • 21 Sep 2017 Ipsen initiates a phase I pharmacokinetics trial in USA (PO) (NCT03302845)
  • 19 Sep 2017 Registered for Malignant carcinoid syndrome (Adjunctive treatment, Treatment-experienced) in Liechtenstein, Iceland, Norway, European Union (PO)
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