Drug Profile


Alternative Names: '761; 2248761 - ViiV Healthcare; GSK2248761; GSK2248761A; IDX-12899; IDX-899

Latest Information Update: 25 Mar 2017

Price : $50

At a glance

  • Originator Idenix Pharmaceuticals
  • Developer GlaxoSmithKline; ViiV Healthcare
  • Class Amides; Antivirals; Indoles; Nitriles; Phosphinic acids; Small molecules
  • Mechanism of Action Non-nucleoside reverse transcriptase inhibitors
  • Orphan Drug Status

    Orphan designation is assigned by a regulatory body to encourage companies to develop drugs for rare diseases.

  • New Molecular Entity Yes

Highest Development Phases

  • Discontinued HIV-1 infections

Most Recent Events

  • 15 Mar 2012 Fosdevirine is no longer licensed to ViiV Healthcare
  • 05 May 2011 GlaxoSmithKline terminates a phase I drug-interaction trial in the USA (NCT01195974)
  • 10 Feb 2011 The US FDA places a clinical hold on GSK 2248761 for the treatment of HIV infections
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