Research programme: thapsigargin analogues - Inspyr Therapeutics

Drug Profile

Research programme: thapsigargin analogues - Inspyr Therapeutics

Alternative Names: Ac-GKAFRR-L12ADT; G-114; G-115; G-301; Plant-derived cytotoxin- Inspyr Therapeutics; Thapsigargin analogues research programme- Inspyr Therapeutics

Latest Information Update: 10 Aug 2016

Price : $50

At a glance

  • Originator GenSpera
  • Developer Inspyr Therapeutics
  • Class Lactones; Peptides; Sesquiterpenes
  • Mechanism of Action Sarcoplasmic reticulum calcium-transporting ATPase inhibitors
  • Orphan Drug Status

    Orphan designation is assigned by a regulatory body to encourage companies to develop drugs for rare diseases.

  • New Molecular Entity No
  • Available For Licensing Yes

Highest Development Phases

  • Preclinical Prostate cancer

Most Recent Events

  • 01 Aug 2016 GenSpera is now called Inspyr Therapeutics
  • 06 May 2015 GenSpera has patents pending for injectable cancer compositions of thapsigargin-containing prodrugs in 17 countries, including Europe, Eurasia, Japan, China, Brazil and USA
  • 29 Apr 2015 GenSpera has patent protection for thapsigargin analogues in USA
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