ARQ 087

Drug Profile

ARQ 087

Alternative Names: ARQ-087

Latest Information Update: 10 Apr 2017

Price : $50

At a glance

  • Originator ArQule
  • Class Antineoplastics; Small molecules
  • Mechanism of Action Fibroblast growth factor receptor antagonists; Phosphotransferase inhibitors
  • Orphan Drug Status

    Orphan designation is assigned by a regulatory body to encourage companies to develop drugs for rare diseases.

    Yes - Cholangiocarcinoma
  • New Molecular Entity Yes

Highest Development Phases

  • Phase II Cholangiocarcinoma
  • Phase I Solid tumours

Most Recent Events

  • 09 Mar 2017 ArQule has patent protection for ARQ 087 in the European Union, Australia, China, Japan, Israel, Taiwan, the Philippines, Mexico, Macau and South Africa (ArQule's form 10-K, filed in March 2015)
  • 08 Mar 2017 ArQule completes enrolment in its phase I/II trial for Cholangiocarcinoma in USA and Italy (NCT01752920)
  • 30 Jun 2016 Preliminary efficacy and adverse events data from a phase I/II trial in Cholangiocarcinoma (Intrahepatic) presented at the 41st European Society for Medical Oncology Congress (ESMO-2016)
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