Drug Profile
Stenoparib - Allarity Therapeutics
Alternative Names: 2X-121; 2X-121/PARPi; E-7449; MGI 25036Latest Information Update: 29 Jun 2023
Price :
$50
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At a glance
- Originator Eisai Co Ltd
- Developer Allarity Therapeutics
- Class Antineoplastics; Antivirals; Isoindoles; Pyridazines; Quinazolines; Small molecules
- Mechanism of Action Poly(ADP-ribose) polymerase 1 inhibitors; Poly(ADP-ribose) polymerase 2 inhibitors; Tankyrase inhibitors
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Orphan Drug Status
Orphan designation is assigned by a regulatory body to encourage companies to develop drugs for rare diseases.
- New Molecular Entity Yes
Highest Development Phases
- Phase II Breast cancer; Ovarian cancer
- Phase I/II Solid tumours
- Preclinical COVID 2019 infections
- No development reported B-cell lymphoma; Neuroblastoma; Renal cancer; Sarcoma
Most Recent Events
- 20 Feb 2023 Phase-I clinical trials in Solid tumours (Monotherapy, Late-stage disease, Second-line therapy or greater) in USA (PO) (NCT05571969)
- 20 Feb 2023 Phase-I clinical trials in Solid tumours (Combination therapy, Late-stage disease, Second-line therapy or greater) in USA (PO) (NCT05571969)
- 09 Dec 2022 Phase-I clinical trials in Ovarian cancer (Second-line therapy or greater, Combination therapy) (PO) prior to December 2022 (Allarity Therapeutics pipeline; December 2022)