GSK 525762

Drug Profile

GSK 525762

Alternative Names: GSK525762

Latest Information Update: 02 Aug 2017

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At a glance

  • Originator GlaxoSmithKline
  • Class Antineoplastics; Benzodiazepines; Small molecules
  • Mechanism of Action Bromodomain and extraterminal domain protein inhibitors
  • Orphan Drug Status

    Orphan designation is assigned by a regulatory body to encourage companies to develop drugs for rare diseases.

  • New Molecular Entity Yes

Highest Development Phases

  • Phase I/II Breast cancer; Carcinoma; Haematological malignancies; Solid tumours
  • Phase I Prostate cancer

Most Recent Events

  • 25 Aug 2017 GlaxoSmithKline plans a phase I/II trial in combination with trametinib for Solid tumours and Small-cell lung cancer (Combination therapy, Late-stage disease, Metastatic disease, Inoperable/Unresectable) (NCT03266159)
  • 31 May 2017 Phase-I clinical trials in Prostate cancer (Combination therapy, Hormone refractory, Metastatic disease, Late-stage disease) in USA (PO) (NCT03150056)
  • 15 May 2017 GlaxoSmithKline plans a phase I trial for Solid tumours (Combination therapy, Second-line therapy or greater, Late-stage disease, Metastatic disease) (NCT03150056)
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