Research programme: GPCR modulators - cancer therapies - Heptares Therapeutics

Drug Profile

Research programme: GPCR modulators - cancer therapies - Heptares Therapeutics

Alternative Names: Adenosine A2A modulators; CXCR-4 modulators

Latest Information Update: 25 May 2016

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At a glance

  • Originator Heptares Therapeutics
  • Developer AstraZeneca; Heptares Therapeutics
  • Class Small molecules
  • Mechanism of Action Adenosine A2A receptor antagonists; Chemokine receptor antagonists; G protein-coupled receptor modulators
  • Orphan Drug Status

    Orphan designation is assigned by a regulatory body to encourage companies to develop drugs for rare diseases.

  • New Molecular Entity Yes

Highest Development Phases

  • Preclinical Cancer

Most Recent Events

  • 25 May 2016 Preclinical trials in Cancer in United Kingdom (PO) before May 2016
  • 23 Feb 2015 Heptares Therapeutics has been acquired by Sosei
  • 15 Dec 2014 Heptares Therapeutics has patent protection for StaR™ (stabilised receptor) technology platform in USA, Europe, China, Japan and Australia
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