Drug Profile
Rupitasertib - Evexta Bio
Alternative Names: DIACC-3010; M-2698; MSC-2363318ALatest Information Update: 24 Apr 2024
Price :
$50
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At a glance
- Originator EMD Serono
- Developer EMD Serono; Evexta Bio
- Class Antineoplastics; Small molecules
- Mechanism of Action 70 kDa ribosomal protein S6 kinase inhibitors; Proto oncogene protein c-akt inhibitors
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Orphan Drug Status
Orphan designation is assigned by a regulatory body to encourage companies to develop drugs for rare diseases.
- New Molecular Entity Yes
Highest Development Phases
- Phase I HER2 positive breast cancer; Solid tumours
- Preclinical Gastric cancer; Glioblastoma; HER2 negative breast cancer
Most Recent Events
- 22 Apr 2024 Preclinical trials in HER2-negative-breast-cancer in France (PO) before April 2024
- 22 Apr 2024 Pharmacodynamics data from preclinical in HER2 negative breast cancer released by Evexta Bio
- 22 Apr 2024 Evexta Bio plans a phase II trial for HER2 negative breast cancer (Combination therapy, Late stage disease) in Q4 in 2024