Drug Profile
APX 3330
Alternative Names: APX-3330; E-3330Latest Information Update: 16 Apr 2024
Price :
$50
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At a glance
- Originator Eisai Co Ltd
- Developer Apexian Pharmaceuticals; Ocuphire Pharma
- Class Anti-inflammatories; Antineoplastics; Antivirals; Eye disorder therapies; Hepatoprotectants; Neuroprotectants; Quinones; Small molecules
- Mechanism of Action Angiogenesis inhibitors; APEX1 protein inhibitors; DNA apurinic apyrimidinic site lyase inhibitors
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Orphan Drug Status
Orphan designation is assigned by a regulatory body to encourage companies to develop drugs for rare diseases.
- New Molecular Entity Yes
- Available For Licensing Yes
Highest Development Phases
- Phase II Diabetic macular oedema; Diabetic retinopathy; Hepatitis B; Hepatitis C; Liver cirrhosis
- Phase I Solid tumours
- Preclinical Inflammatory bowel diseases; Pancreatic cancer
- Discontinued Haematological malignancies; Liver disorders; Peripheral nervous system diseases
Most Recent Events
- 16 Apr 2024 Discontinued - Phase-I for Peripheral nervous system diseases (Chemotherapy-induced) in USA (PO) before April 2024 (Apexian Pharmaceuticals pipeline, April 2024)
- 29 Feb 2024 Ocuphire Pharma files special protocol assessment (SPA) to US FDA for phase-III trial for Diabetic retinopathy
- 02 Nov 2023 Ocuphire Pharma announces successful End-of-Phase II Meeting with US FDA for APX 3330 in Diabetic Retinopathy