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Gabapentin enacarbil

Drug Profile

Gabapentin enacarbil

Alternative Names: 1838262; ASP8825; Gabapentin-XP; GSK 1838262; Horizant; Regnite; Solzira; XP13512

Latest Information Update: 04 Nov 2018

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At a glance

  • Originator XenoPort
  • Developer Arbor Pharmaceuticals; Astellas Pharma; GlaxoSmithKline; National Institute on Alcohol Abuse and Alcoholism; XenoPort
  • Class Acetic acids; Antiepileptic drugs; Carbamates; Cyclohexanecarboxylic acids; Small molecules
  • Mechanism of Action CACNA2D1 protein modulators; GABA receptor agonists
  • Orphan Drug Status

    Orphan designation is assigned by a regulatory body to encourage companies to develop drugs for rare diseases.

  • New Molecular Entity Yes
  • Available For Licensing Yes - Restless legs syndrome

Highest Development Phases

  • Marketed Postherpetic neuralgia; Restless legs syndrome
  • Phase II Alcoholism
  • Discontinued Diabetic neuropathies; Migraine

Most Recent Events

  • 24 Jun 2018 Biomarkers information updated
  • 19 Jul 2017 XenoPort terminates a phase I trial in Restless legs syndrome (In adolescents) in USA, due to lack of enrolment (PO) (NCT02633657)
  • 01 Mar 2017 XenoPort completes the phase II trial in Alcoholism in USA (PO) (NCT02252536)
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