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Telotristat etiprate - TerSera Therapeutics

Drug Profile

Telotristat etiprate - TerSera Therapeutics

Alternative Names: LP-778914; LX-1032; LX-1606; LX1032 hippurate; LX1606 hippurate; Telotristat ethyl; Xermelo

Latest Information Update: 11 Mar 2024

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At a glance

  • Originator Lexicon Pharmaceuticals
  • Developer Ipsen; Lexicon Pharmaceuticals
  • Class Amines; Anti-inflammatories; Antineoplastics; Chlorobenzenes; Fluorinated hydrocarbons; Propionic acids; Pyrazoles; Pyrimidines; Small molecules
  • Mechanism of Action Tryptophan hydroxylase inhibitors
  • Orphan Drug Status

    Orphan designation is assigned by a regulatory body to encourage companies to develop drugs for rare diseases.

    Yes - Malignant carcinoid syndrome
  • New Molecular Entity Yes

Highest Development Phases

  • Marketed Malignant carcinoid syndrome
  • Phase II Neuroendocrine tumours
  • Preclinical Cholangiocarcinoma; Colorectal cancer; Liposarcoma
  • Discontinued Biliary cancer; Ulcerative colitis

Most Recent Events

  • 18 Jan 2024 Efficacy and adverse events data from a phase II trial in Biliary tract cancer presented at the 2024 Gastrointestinal Cancers Symposium (ASCO-GCS-2024)
  • 21 Feb 2023 TerSera Therapeutics and University of Kentucky terminates a phase-II clinical trials in Neuroendocrine tumours (In adults, In the elderly, Metastatic disease, Inoperable/Unresectable, Second-line therapy or greater, Combination therapy) in USA (PO, Tablet) as sponsor cancelled research (NCT04543955)
  • 05 May 2022 Novartis suspends a phase II trial in Neuroendocrine tumours (In adults, In the elderly, Metastatic disease, Inoperable/Unresectable, Second-line therapy or greater, Combination therapy) in USA (PO) due to production suspension of Lutathera (NCT04543955)
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