EZN 3042
Alternative Names: EZN-3042; SPC 3042Latest Information Update: 17 Jan 2024
At a glance
- Originator Santaris Pharma
- Developer Enzon Pharmaceuticals; Roche
- Class Antineoplastics; Antisense oligonucleotides
- Mechanism of Action BIRC5 protein inhibitors
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Orphan Drug Status
Orphan designation is assigned by a regulatory body to encourage companies to develop drugs for rare diseases.
- New Molecular Entity Yes
Highest Development Phases
- Phase I Lymphoma; Precursor cell lymphoblastic leukaemia-lymphoma; Solid tumours
Most Recent Events
- 17 Jan 2024 EZN 3042 is still in phase-I trial for Lymphoma, Precursor cell lymphoblastic leukaemia-lymphoma (In children) and Solid tumours in Australia, Brazil, Canada, France, USA (Enzon Pharmaceuticals pipeline, January 2024)
- 07 Mar 2012 Discontinued - Phase-I for Acute lymphoblastic leukaemia in Australia (IV)
- 07 Mar 2012 Discontinued - Phase-I for Acute lymphoblastic leukaemia in Brazil (IV)