Cenerimod - Idorsia Pharmaceuticals
Alternative Names: ACT-334441; Second selective S1P1 receptor agonist - IdorsiaLatest Information Update: 10 Apr 2026
At a glance
- Originator Actelion Pharmaceuticals
- Developer Idorsia Pharmaceuticals; Viatris
- Class Antirheumatics; Oxadiazoles; Pyridines; Small molecules
- Mechanism of Action Sphingosine 1 phosphate receptor modulators
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Orphan Drug Status
No
Orphan designation is assigned by a regulatory body to encourage companies to develop drugs for rare diseases.
- New Molecular Entity Yes
Highest Development Phases
- Phase III Lupus nephritis; Systemic lupus erythematosus
- Phase I Unspecified
- Preclinical Rheumatoid arthritis
- No development reported Autoimmune disorders
Most Recent Events
- 18 Mar 2026 Viatris completes a phase-I Bioavailability trial (In volunteers) in Netherlands (PO, IV), (NCT07301723)
- 12 Dec 2025 Phase-II clinical trials in Systemic lupus erythematosus (Adjunctive treatment) in China (PO) (NCT07266090)
- 11 Dec 2025 Phase-I clinical trials in Unspecified (In volunteers) in Netherlands (IV, Infusion), (NCT07301723)