Drug Profile
Research programme: histone methyltransferase inhibitors - Epizyme
Alternative Names: CARM1 inhibitors; coactivator-associated arginine methyltransferase 1 inhibitors; EPZ 020411; HMT 2; HMT 3; HMT inhibitors; PRMT1 inhibitors; PRMT3 inhibitors; PRMT6 inhibitors; PRMT8 inhibitors; Protein arginine methyltransferase 1 inhibitors; Protein arginine methyltransferase 3 inhibitors; Protein arginine methyltransferase 6 inhibitors; Protein arginine methyltransferase 8 inhibitorsLatest Information Update: 17 Oct 2022
Price :
$50
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At a glance
- Originator Epizyme
- Developer Celgene International SARL; Epizyme
- Class Antineoplastics; Pyrazoles
- Mechanism of Action Histone methyltransferase inhibitors
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Orphan Drug Status
Orphan designation is assigned by a regulatory body to encourage companies to develop drugs for rare diseases.
- New Molecular Entity Yes
Highest Development Phases
- Preclinical Haematological malignancies; Solid tumours
Most Recent Events
- 14 Oct 2022 Research programme: histone methyltransferase inhibitors is still in preclinical trials for Haematological malignancies in USA (Epizyme pipeline, October 2022)
- 14 Oct 2022 Research programme: histone methyltransferase inhibitors is still in preclinical trials for Solid tumours in USA (Epizyme pipeline, October 2022)
- 12 Aug 2022 Epizyme has been acquired by Ipsen