Bromopyruvate - PreScience Labs
Alternative Names: 3-bromopyruvate; 3-bromopyruvic acid; 3-BrPA; 3BP; KAT 3-BP; KAT-101; KAT-201; KAT/3BP; PSL-001Latest Information Update: 23 Jun 2025
At a glance
- Originator Johns Hopkins University
- Developer NewG Lab; PreScience Labs
- Class Antineoplastics; Keto acids; Pyruvates; Small molecules
- Mechanism of Action Alkylating agents; MASP2 protein inhibitors; Pyruvate dehydrogenase complex inhibitors
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Orphan Drug Status
Orphan designation is assigned by a regulatory body to encourage companies to develop drugs for rare diseases.
- New Molecular Entity Yes
Highest Development Phases
- Phase I/II Pancreatic cancer
- Preclinical Lymphoma
- Discontinued Cancer
Most Recent Events
- 05 Jun 2025 Primocure Pharma suspends a phase I/II trial in Pancreatic cancer (Inoperable/Unresectable, Late-stage disease, Metastatic disease) in South Korea (Intratumoural, PO) due to enrolment pause
- 20 Dec 2023 Discontinued - Preclinical for Cancer in USA (Intra-arterial)
- 20 Dec 2023 Pharmacodynamics data from preclinical studies in Pancreatic cancer released by PrimoCure Pharma (PrimoCure Pharma pipeline, December 2023)