Rupitasertib - Evexta Bio
Alternative Names: DIACC-3010; M-2698; MSC-2363318ALatest Information Update: 28 Jun 2025
At a glance
- Originator EMD Serono
- Developer EMD Serono; Evexta Bio
- Class Antineoplastics; Small molecules
- Mechanism of Action 70 kDa ribosomal protein S6 kinase inhibitors; Proto-oncogene protein c-akt inhibitors
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Orphan Drug Status
Orphan designation is assigned by a regulatory body to encourage companies to develop drugs for rare diseases.
- New Molecular Entity Yes
Highest Development Phases
- Preclinical Gastric cancer; Glioblastoma; HER2 negative breast cancer
- No development reported HER2 positive breast cancer; Solid tumours
Most Recent Events
- 28 Jun 2025 No recent reports of development identified for phase-I development in HER2-positive-breast-cancer(Combination therapy, Late-stage disease, Metastatic disease) in USA (PO)
- 28 Jun 2025 No recent reports of development identified for phase-I development in Solid-tumours(Combination therapy, Late-stage disease) in USA (PO)
- 28 Jun 2025 No recent reports of development identified for phase-I development in Solid-tumours(Late-stage disease, Monotherapy) in USA (PO)