TAK 243
Alternative Names: AOB-87172; MLN-7243; TAK-243Latest Information Update: 28 Jan 2025
At a glance
- Originator Millennium
- Developer Takeda Oncology
- Class Antineoplastics; Cyclopentanes; Organic sulfur compounds; Pyrazoles; Pyrimidines; Small molecules
- Mechanism of Action NF-kappa B inhibitors; Ubiquitin protein ligase inhibitors
-
Orphan Drug Status
Orphan designation is assigned by a regulatory body to encourage companies to develop drugs for rare diseases.
- New Molecular Entity Yes
Highest Development Phases
- Preclinical Lymphoma
- No development reported Acute myeloid leukaemia; Chronic lymphocytic leukaemia; Diffuse large B cell lymphoma; Solid tumours
Most Recent Events
- 28 Jan 2025 No recent reports of development identified for phase-I development in Solid-tumours(Late-stage disease, Second-line therapy or greater) in USA (IV, Infusion)
- 28 Jan 2025 No recent reports of development identified for preclinical development in Acute-myeloid-leukaemia in USA (IV, Infusion)
- 28 Jan 2025 No recent reports of development identified for preclinical development in Chronic-lymphocytic-leukaemia in USA (IV)