Tasurgratinib succinate - Eisai Co Ltd
Alternative Names: E-7090; TASFYGOLatest Information Update: 11 Mar 2025
At a glance
- Originator Eisai Co Ltd
- Class Amides; Amines; Antineoplastics; Benzene derivatives; Ethers; Indoles; Piperidines; Pyridines; Small molecules
- Mechanism of Action Type 1 fibroblast growth factor receptor antagonists; Type 3 fibroblast growth factor receptor antagonists; Type-2 fibroblast growth factor receptor antagonists
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Orphan Drug Status
Orphan designation is assigned by a regulatory body to encourage companies to develop drugs for rare diseases.
- New Molecular Entity Yes
Highest Development Phases
- Marketed Biliary cancer
- Phase II Cholangiocarcinoma; Solid tumours
- Phase I HER2 negative breast cancer
Most Recent Events
- 28 Feb 2025 Tasurgratinib succinate licensed to Sciclone Pharmaceuticals in China, Hong Kong, Macau, Taiwan
- 10 Dec 2024 Efficacy data from a phase I trial in Breast cancer was presented at the 47th Annual San Antonio Breast Cancer Symposium (SABCS-2024)
- 20 Nov 2024 Launched for Biliary cancer (Inoperable/Unresectable, Metastatic disease, Late-stage disease, Second-line therapy or greater) in Japan (PO) - First global launch