Brepocitinib - Priovant Therapeutics
Alternative Names: Brepocitinib tosylate - Pfizer; PF 6700841; PF-06700841; PF-06700841-15; PF-841Latest Information Update: 23 Sep 2025
At a glance
- Originator Pfizer
- Developer Pfizer; Priovant Therapeutics
- Class Amides; Anti-inflammatories; Antipsoriatics; Antirheumatics; Arylsulfonic acids; Bridged-ring heterocyclic compounds; Cyclopropanes; Fluorinated hydrocarbons; Ketones; Pyrazoles; Pyrimidines; Skin disorder therapies; Small molecules
- Mechanism of Action Janus kinase 1 inhibitors; TYK2 kinase inhibitors
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Orphan Drug Status
Orphan designation is assigned by a regulatory body to encourage companies to develop drugs for rare diseases.
- New Molecular Entity Yes
Highest Development Phases
- Phase III Dermatomyositis; Uveitis
- Phase II Crohn's disease; Hidradenitis suppurativa; Sarcoidosis
- Discontinued Alopecia; Alopecia areata; Atopic dermatitis; Lupus vulgaris; Plaque psoriasis; Psoriatic arthritis; Systemic lupus erythematosus; Ulcerative colitis; Vitiligo
Most Recent Events
- 17 Sep 2025 Efficacy and adverse events data from a phase III VALOR trial in dermatomyositis released by Priovant
- 17 Sep 2025 Priovant plans to file an NDA for brepocitinib in dermatomyositis in the first half of 2026
- 09 Apr 2025 Phase-II BEACON clinical trials in Sarcoidosis in USA (PO) (NCT06978725)