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Research programme: bromodomain and extraterminal domain protein inhibitors - Checkpoint Therapeutics

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Drug Profile

Research programme: bromodomain and extraterminal domain protein inhibitors - Checkpoint Therapeutics

Alternative Names: BET inhibitors; BRD4 Inhibitors

Latest Information Update: 10 Jun 2025

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At a glance

  • Originator Jubilant Biosys
  • Developer Checkpoint Therapeutics; Jubilant Biosys; TG Therapeutics Inc
  • Class Antineoplastics; Small molecules
  • Mechanism of Action BRD4 protein inhibitors; Bromodomain and extraterminal domain protein inhibitors
  • Orphan Drug Status

    Orphan designation is assigned by a regulatory body to encourage companies to develop drugs for rare diseases.

    No
  • New Molecular Entity Yes

Highest Development Phases

  • No development reported Cancer

Most Recent Events

  • 30 May 2025 Checkpoint Therapeutics has been acquired by Sun Pharmaceutical Industries
  • 28 Mar 2024 No recent reports of development identified for preclinical development in Cancer in USA
  • 16 Mar 2022 Preclinical development is still ongoing in Cancer in USA (Jubilant Therapeutics pipeline, March 2022)

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