Dapolsertib - Menarini
Alternative Names: MEN 1703; MEN1703/SEL24; SEL 24; SEL24 program; SEL24-1; SEL24-B489; SEL24/MEN1703Latest Information Update: 06 May 2025
At a glance
- Originator Selvita
- Developer Menarini; Ryvu Therapeutics; Theradex
- Class Antineoplastics; Benzimidazoles; Halogenated hydrocarbons; Nitro compounds; Small molecules
- Mechanism of Action Fms-like tyrosine kinase 3 inhibitors; Proto oncogene protein c pim 1 inhibitors
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Orphan Drug Status
Orphan designation is assigned by a regulatory body to encourage companies to develop drugs for rare diseases.
- New Molecular Entity Yes
Highest Development Phases
- Phase II Acute myeloid leukaemia; B-cell lymphoma; Diffuse large B cell lymphoma
- Preclinical Myelofibrosis
Most Recent Events
- 25 Apr 2025 Phase-II clinical trials in Diffuse large B cell lymphoma (Combination therapy, Second-line therapy or greater) in France (PO) (NCT06534437) (Ryvu Therapeutics pipeline, May 2025)
- 25 Apr 2025 Phase-II clinical trials in Diffuse large B cell lymphoma (Combination therapy, Second-line therapy or greater) in Spain (PO) (NCT06534437) (Ryvu Therapeutics pipeline, May 2025)
- 25 Apr 2025 Phase-II clinical trials in Diffuse large B cell lymphoma (Second-line therapy or greater, Monotherapy) in France (PO) (NCT06534437) (Ryvu Therapeutics pipeline, May 2025)