Drug Profile
Tegatrabetan
Alternative Names: BC-2059Latest Information Update: 12 Apr 2017
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At a glance
- Originator BetaCat Pharmaceuticals
- Class Antineoplastics; Small molecules
- Mechanism of Action Beta catenin inhibitors; Wnt signalling pathway inhibitors
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Orphan Drug Status
Orphan designation is assigned by a regulatory body to encourage companies to develop drugs for rare diseases.
- New Molecular Entity Yes
Highest Development Phases
- Preclinical Acute myeloid leukaemia; Fibroma; Multiple myeloma
Most Recent Events
- 13 Mar 2018 Beta Cat Pharmaceuticals plans a phase I trial for Fibroma (Recurrent, Inoperable/unresectable, Second-line therapy or greater) in March 2018 (NCT03459469)
- 12 Apr 2017 BetaCat Pharmaceuticals has patents pending for transducin β-like protein 1 inhibitors in European Union, Eastern Europe, India, China, Japan, and Canada
- 12 Apr 2017 BetaCat Pharmaceuticals has patent protection for transducin β-like protein 1 inhibitors in South Korea, Mexico, New Zealand, Singapore, South Africa, Eurasia