Buprenorphine oral lyophilisates
Alternative Names: buprenorphine hydrochloride; EspranorLatest Information Update: 13 Jan 2022
Price :
$50 *
At a glance
- Originator Martindale Pharmaceuticals
- Class Cyclopropanes; Drug withdrawal therapies; Morphinans; Opioid analgesics; Small molecules
- Mechanism of Action Nociceptin receptor agonists; Opioid delta receptor agonists; Opioid kappa receptor antagonists; Opioid mu receptor agonists
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Orphan Drug Status
Orphan designation is assigned by a regulatory body to encourage companies to develop drugs for rare diseases.
- New Molecular Entity No
Highest Development Phases
- Marketed Opioid-related disorders
Most Recent Events
- 19 Jun 2017 Chemical structure information added
- 05 May 2017 Scottish Medicines Consortium is reviewing oral lyophilisates of buprenorphine for use in Scotland
- 05 May 2017 Interim adverse events, pharmacokinetics, pharmacodynamics data from a phase II trial in Opioid abuse released by Martindale Pharmaceuticals