Certepetide - Lisata Therapeutics
Alternative Names: CEND-1; Internalised-arginylglycylaspartic Acid Cyclic Peptide; iRGD; LSTA-1; QLC-12102Latest Information Update: 21 Jul 2025
At a glance
- Originator DrugCendR
- Developer Australasian Gastro-Intestinal Trials Group; Lisata Therapeutics; National Health and Medical Research Council Clinical Trials Centre; Qilu Pharmaceutical; The University of Kansas Cancer Center; University of Sydney
- Class Antineoplastics; Cyclic peptides; Peptides
- Mechanism of Action Integrin alphaV antagonists; Neuropilin-1 stimulants
-
Orphan Drug Status
Orphan designation is assigned by a regulatory body to encourage companies to develop drugs for rare diseases.
- New Molecular Entity Yes
- Available For Licensing Yes
Highest Development Phases
- Phase II Adenocarcinoma; Glioblastoma; Pancreatic cancer; Solid tumours
- Phase I/II Colorectal cancer; Gastrointestinal cancer
Most Recent Events
- 17 Jul 2025 Updated efficacy data from the phase Ib/IIa iLSTA trial in Pancreatic cancer released by Lisata Therapeutics
- 17 Jul 2025 Lisata Therapeutics completes enrolment in the phase I/II iLSTA trial in Pancreatic cancer (First-line therapy, Combination therapy, Late-stage disease, Metastatic disease, Inoperable/Unresectable) in Australia (IV) (ACTRN12623000223639)
- 16 Jul 2025 Lisata Therapeutics has patent protection for 'composition of matter' in USA