ASTX 029
Alternative Names: ASTX-029Latest Information Update: 05 May 2025
At a glance
- Originator Astex Pharmaceuticals
- Class Amides; Amines; Antineoplastics; Halogenated hydrocarbons; Phenyl ethers; Pyrans; Pyrimidines; Small molecules
- Mechanism of Action Mitogen-activated protein kinase 1 inhibitors; Mitogen-activated protein kinase 3 inhibitors
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Orphan Drug Status
Orphan designation is assigned by a regulatory body to encourage companies to develop drugs for rare diseases.
- New Molecular Entity Yes
Highest Development Phases
- Phase I/II Solid tumours
- Preclinical Acute myeloid leukaemia; Uveal melanoma
Most Recent Events
- 05 May 2025 Mosaic Therapeutics in-licenses ASTX 029 from Astex Pharmaceuticals
- 24 Apr 2025 Astex Pharmaceuticals plans a clinical trial for Cancer (Combination-therapy) in 2026
- 20 Feb 2025 Pharmacodynamics data from a preclinical trial in Acute-myeloid leukaemia presented at 66th American Society of Hematology Annual Meeting and Exposition 2024 (ASH-Hem-2024)