Sirolimus - Emtora Biosciences
Alternative Names: Encapsulated rapamycin; Encapsulated rapamycin - Emtora Biosciences; eRapa™; MTX-230Latest Information Update: 22 Sep 2026
At a glance
- Originator University of Texas Health Science Center at San Antonio
- Developer Biodexa Pharmaceuticals; Emtora Biosciences
- Class 3-ring heterocyclic compounds; Alcohols; Alkenes; Anti-infectives; Anti-inflammatories; Antiepileptic drugs; Antifungals; Antineoplastics; Aza compounds; Cardiovascular therapies; Cyclic ethers; Cyclohexanols; Esters; Eye disorder therapies; Ketones; Lactones; Macrocyclic compounds; Macrolides; Methyl ethers; Nootropics; Piperidines; Polyenes; Pyridines; Skin disorder therapies
- Mechanism of Action Immunosuppressants; Methylmalonyl CoA mutase stimulants; MTOR protein inhibitors; T lymphocyte inhibitors
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Orphan Drug Status
Yes - Familial adenomatous polyposis
Orphan designation is assigned by a regulatory body to encourage companies to develop drugs for rare diseases.
- New Molecular Entity No
Highest Development Phases
- Phase III Familial adenomatous polyposis
- Phase II Bladder cancer
- No development reported Autoimmune disorders; Breast cancer; Cognition disorders; Lung cancer; Prostate cancer
Most Recent Events
- 14 Sep 2026 Emtora Biosciences completes enrolment in phase-II clinical trials in Bladder cancer in USA (PO) (NCT04375813)
- 28 Aug 2026 No recent reports of development identified for phase-I development in Prostate-cancer(Early-stage disease) in USA (PO, Capsule)
- 21 Aug 2026 Phase-III clinical trials in Familial adenomatous polyposis in Italy (PO)