Research programme: pyrazolopyrimidine derivatives - Lead Discovery Siena
Latest Information Update: 28 Oct 2022
At a glance
- Originator University of Siena
- Developer Lead Discovery Siena
- Class Antineoplastics; Pyrazoles; Pyrimidines; Small molecules
- Mechanism of Action Src-family kinase inhibitors
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Orphan Drug Status
Orphan designation is assigned by a regulatory body to encourage companies to develop drugs for rare diseases.
- New Molecular Entity Yes
- Available For Licensing Yes - Cancer; Glioblastoma
Highest Development Phases
- No development reported Glioblastoma
Most Recent Events
- 28 Oct 2022 No recent reports of development identified for preclinical development in Glioblastoma in Italy (Parenteral)
- 05 Sep 2018 Pyrazolopyrimidine derivatives - Lead Discovery Siena is available for licensing as of 05 Sep 2018. http://leaddiscoverysiena.it/about-us/ (Lead Discovery Siena website, September 2018)
- 05 Sep 2018 Preclinical trials in Glioblastoma in Italy (Parenteral) (Lead Discovery Siena Pipeline, September 2018)