Research programme: SETD2 inhibitors - Epizyme
Alternative Names: EPZ-040414Latest Information Update: 28 Jan 2023
At a glance
- Originator Epizyme
- Class Antineoplastics; Small molecules
- Mechanism of Action Histone-lysine N-methyltransferase inhibitors
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Orphan Drug Status
Orphan designation is assigned by a regulatory body to encourage companies to develop drugs for rare diseases.
- New Molecular Entity Yes
Highest Development Phases
- No development reported Multiple myeloma