Emzadirib - Cyteir Therapeutics
Alternative Names: CYT-0851Latest Information Update: 23 Sep 2025
At a glance
- Originator Cyteir Therapeutics
- Class Anilides; Antineoplastics; Carbamates; Cyclohexanes; Small molecules; Sulfonamides; Thiazoles
- Mechanism of Action Monocarboxylic acid transporter inhibitors; Rad51 recombinase inhibitors
-
Orphan Drug Status
No
Orphan designation is assigned by a regulatory body to encourage companies to develop drugs for rare diseases.
- New Molecular Entity Yes
Highest Development Phases
- Discontinued Haematological malignancies; Solid tumours
Most Recent Events
- 23 Sep 2025 Chemical structure information added.
- 20 Dec 2024 Cyteir Therapeutics completes a phase I/II trial for Solid tumours and B-cell malignancies (Monotherapy, Combination therapy, Second line therapy or greater, Metastatic disease, Recurrent, Late-stage disease) in USA (PO) (NCT03997968)
- 20 Mar 2024 Cyteir Therapeutics winds down its business and remains no longer active (Cyteir Therapeutic pipeline, May 2024)