Vipoglanstat - Gesynta Pharma
Alternative Names: BI-1029539; GS-248; OX-MPILatest Information Update: 23 Mar 2026
At a glance
- Originator Biolipox
- Developer Gesynta Pharma
- Class Anti-inflammatories; Skin disorder therapies; Small molecules; Vascular disorder therapies; Vasodilators
- Mechanism of Action Prostaglandin-E synthase inhibitors
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Orphan Drug Status
Yes - Systemic scleroderma
Orphan designation is assigned by a regulatory body to encourage companies to develop drugs for rare diseases.
- New Molecular Entity Yes
- Available For Licensing Yes
Highest Development Phases
- Phase II Endometriosis; Systemic scleroderma
Most Recent Events
- 11 Mar 2026 Pharmacodynamics data from a preclinical studies in Endometriosis released by Gesynta Pharma
- 15 Oct 2025 Phase-II clinical trials in Endometriosis in Italy, Poland, Romania, Bulgaria, Czech Republic, Hungary (PO) (NCT07260669)
- 15 Oct 2025 Phase-II clinical trials in Endometriosis (In adults) in United Kingdom (PO) (NCT07260669)