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Lunresertib - Repare Therapeutics

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Drug Profile

Lunresertib - Repare Therapeutics

Alternative Names: CCNE1-SL inhibitor - Repare Therapeutics; Lunre; Manchester; RP-6306

Latest Information Update: 24 Jun 2025

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At a glance

  • Originator Repare Therapeutics
  • Developer Canadian Cancer Trials Group; Repare Therapeutics; University Health Network
  • Class Amides; Antineoplastics; Pyridines; Small molecules
  • Mechanism of Action PKMYT1 protein inhibitors
  • Orphan Drug Status

    Orphan designation is assigned by a regulatory body to encourage companies to develop drugs for rare diseases.

    No
  • New Molecular Entity Yes
  • Available For Licensing Yes

Highest Development Phases

  • Phase II Solid tumours
  • Phase I Ovarian cancer; Uterine cancer

Most Recent Events

  • 25 Apr 2025 Pharmacodynamics data from a preclinical trial in Breast cancer presented at the 116th Annual Meeting of the American Association for Cancer Research 2025 (AACR-2025)
  • 03 Mar 2025 Lunresertib - Repare Therapeutics is available for licensing as of 03 Mar 2025. http://www.reparerx.com
  • 28 Jan 2025 No recent reports of development identified for phase-I development in Solid-tumours(Combination therapy, Late-stage disease, Metastatic disease, Second-line therapy or greater) in United Kingdom (PO, Capsule)

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