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Azenosertib - Zentalis Pharmaceuticals

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Drug Profile

Azenosertib - Zentalis Pharmaceuticals

Alternative Names: KP-2638; ZN-c3

Latest Information Update: 28 May 2025

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At a glance

  • Originator Zentalis Pharmaceuticals
  • Developer GSK; K-Group Beta; Zentalis Pharmaceuticals; Zentera Therapeutics
  • Class Amines; Antineoplastics; Cyclopentanes; Piperazines; Pyrazoles; Pyridines; Pyrimidinones; Small molecules
  • Mechanism of Action WEE1 protein inhibitors
  • Orphan Drug Status

    Orphan designation is assigned by a regulatory body to encourage companies to develop drugs for rare diseases.

    Yes - Osteosarcoma
  • New Molecular Entity Yes

Highest Development Phases

  • Phase II Pancreatic cancer; Solid tumours; Uterine cancer
  • Phase I/II Acute myeloid leukaemia; Colorectal cancer; Fallopian tube cancer; Osteosarcoma; Ovarian cancer; Peritoneal cancer; Triple negative breast cancer
  • Phase I Breast cancer

Most Recent Events

  • 28 May 2025 No recent reports of development identified for phase-I development in Ovarian-cancer(Combination therapy, In the elderly, Second-line therapy or greater, In adults) in Serbia (PO)
  • 14 May 2025 Efficacy data from a phase II DENALI trial in Ovarian cancer released by Zentalis Pharmaceuticals
  • 15 Mar 2025 Zentalis Pharmaceuticals plans the phase II DENALI Part 2 trial for Ovarian cancer (PO), in 1H 2025

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