Cannabidiol/tetramethylpyrazine - Artelo Biosciences
Alternative Names: ART-1211; ART12.11; CBD Cocrystal; Tetramethylpyrazine/cannabidiol- Artelo BiosciencesLatest Information Update: 24 Nov 2025
At a glance
- Originator Artelo Biosciences
- Class Alkaloids; Analgesics; Anti-inflammatories; Anti-ischaemics; Antiacnes; Antibacterials; Antidepressants; Antiepileptic drugs; Antihyperglycaemics; Antihyperlipidaemics; Antineoplastics; Antiparkinsonians; Antipsoriatics; Antipsychotics; Antirheumatics; Anxiolytics; Behavioural disorder therapies; Cannabinoids; Cardiovascular therapies; Cyclohexenes; Drug withdrawal therapies; Heart failure therapies; Hepatoprotectants; Muscle relaxants; Neuroprotectants; Obesity therapies; Resorcinols; Skin disorder therapies; Small molecules; Vascular disorder therapies; Vasodilators
- Mechanism of Action 5-HT1 serotonin receptor modulators; Cannabinoid receptor CB1 inverse agonists; Cannabinoid receptor CB2 inverse agonists
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Orphan Drug Status
No
Orphan designation is assigned by a regulatory body to encourage companies to develop drugs for rare diseases.
- New Molecular Entity No
Highest Development Phases
- Preclinical Anxiety disorders; Depressive disorders
- Discontinued Cancer; Inflammatory bowel diseases; Post-traumatic stress disorders; Stroke
Most Recent Events
- 18 Nov 2025 Artelo Biosciences plans a phase I trial for Anxiety disorders and Depressive diorders (PO) in first half of 2026
- 27 Oct 2025 Discontinued - Preclinical for Cancer in USA (PO), before October 2025 (Artelo Biosciences pipeline, June 2022)
- 27 Oct 2025 Discontinued - Preclinical for Inflammatory bowel diseases in USA (PO), before October 2025 (Artelo Biosciences pipeline, October 2025)