Research programme: kt 3000 HDAC and PARP inhibitors - Rakovina Therapeutics
Alternative Names: kt 3000 dual action DNA Damage Response inhibitors - Rakovina Therapeutics; kt-3000; kt-3000 seriesLatest Information Update: 28 Dec 2025
At a glance
- Originator Rakovina Therapeutics
- Developer Rakovina Therapeutics; University of British Columbia
- Class Antineoplastics; Small molecules
- Mechanism of Action DNA repair inhibitors; Histone deacetylase inhibitors; Poly(ADP-ribose) polymerase inhibitors
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Orphan Drug Status
No
Orphan designation is assigned by a regulatory body to encourage companies to develop drugs for rare diseases.
- New Molecular Entity Yes
Highest Development Phases
- No development reported Cancer; Ewing's sarcoma
Most Recent Events
- 28 Dec 2025 No recent reports of development identified for preclinical development in Ewing's Sarcoma in Canada
- 28 May 2025 No recent reports of development identified for preclinical development in Cancer in Canada
- 28 Nov 2023 Rakovina Therapeutics plans to initiate clinical trials for Ewing's sarcoma, in 2024