Drug Profile

Olomorasib - Eli Lilly and Company

Alternative Names: KRAS-G12C-II; LY-3537982

Latest Information Update: 06 Apr 2026

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At a glance

Originator Eli Lilly and Company
Class Antineoplastics; Small molecules
Mechanism of Action KRAS protein inhibitors

Orphan Drug Status

Orphan designation is assigned by a regulatory body to encourage companies to develop drugs for rare diseases.

No
New Molecular Entity Yes

Highest Development Phases

Phase III Non-small cell lung cancer
Phase I Solid tumours

Most Recent Events

06 Apr 2026 3926409 - KDM, DT, HE, TT
02 Mar 2026 Eli Lilly and Company initiates enrolment in a phase I pharmacokinetic trial (In volunteers) in the USA (NCT07439250)
27 Feb 2026 Eli Lilly and Company plans a phase I trial (In volunteers) in USA (PO) in March 2026 (NCT07439250)

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