BBO 10203
Alternative Names: BBO-10203; PI3K alpha:RAS breaker - BridgeBio PharmaLatest Information Update: 19 Dec 2025
At a glance
- Originator BridgeBio Pharma
- Developer BridgeBio Oncology Therapeutics
- Class Antineoplastics; Small molecules
- Mechanism of Action Phosphatidylinositol 3 kinase alpha inhibitors; Ras signal transduction pathway inhibitors
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Orphan Drug Status
No
Orphan designation is assigned by a regulatory body to encourage companies to develop drugs for rare diseases.
- New Molecular Entity Yes
Highest Development Phases
- Phase I Solid tumours
Most Recent Events
- 11 Dec 2025 Pharmacodynamics data from a preclinical trial in Solid tumours released by BridgeBio Oncology Therapeutics
- 28 Nov 2025 Chemical structure information added.
- 25 Oct 2025 Pharmacodynamics and adverse events data from a preclinical trial in Solid tumours released by BridgeBio Oncology Therapeutics