Research programme: casein kinase 1 inhibitors - CasInvent Pharma
Alternative Names: CS1 inhibitors - CasInvent PharmaLatest Information Update: 24 Jun 2025
At a glance
- Originator Masaryk University
- Developer CasInvent Pharma
- Class Antineoplastics; Imidazoles; Pyridines; Pyrroles; Small molecules
- Mechanism of Action Casein kinase I inhibitors; Casein kinase Ialpha inhibitors
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Orphan Drug Status
Orphan designation is assigned by a regulatory body to encourage companies to develop drugs for rare diseases.
- New Molecular Entity Yes
Highest Development Phases
- Preclinical Acute myeloid leukaemia
- Research Colorectal cancer; Malignant melanoma; Pancreatic cancer; Triple negative breast cancer
Most Recent Events
- 25 Apr 2025 Preclinical trials in Acute myeloid leukaemia in Czech Republic (unspecified route), before April 2025
- 25 Apr 2025 Pharmacodynamics and adverse events data from a preclinical trial in Acute myeloid leukemia and Pancreatic cancer presented at the 116th Annual Meeting of the American Association for Cancer Research (AACR-2025)
- 24 Apr 2024 Early research in Colorectal cancer in Czech Republic (unspecified route) (CasInvent Pharma pipeline, April 2024)