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ENDOPIN - BTB Therapeutics

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Drug Profile

ENDOPIN - BTB Therapeutics

Alternative Names: BTB-101

Latest Information Update: 17 Jul 2025

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At a glance

  • Originator Kyoto University
  • Developer BTB Therapeutics; Kyoto University
  • Class Non-opioid analgesics; Small molecules
  • Mechanism of Action Alpha 2b adrenergic receptor antagonists
  • Orphan Drug Status

    Orphan designation is assigned by a regulatory body to encourage companies to develop drugs for rare diseases.

    No
  • New Molecular Entity Yes

Highest Development Phases

  • Phase I/II Postoperative pain
  • Preclinical Cancer pain; Pruritus

Most Recent Events

  • 17 Jul 2025 Preclinical trials in Cancer pain in Japan (PO) prior to July 2025 (BTB Therapeutics pipeline, July 2025)
  • 17 Jul 2025 Preclinical trials in Pruritus in Japan (PO) prior July 2025 (BTB Therapeutics pipeline, July 2025)
  • 24 Apr 2024 Adverse events data from phase I/II trial in Postoperative pain released by Kyoto University

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