BY 101298
Alternative Names: AMO-959; BY-101298; BY-1298Latest Information Update: 19 Dec 2025
At a glance
- Originator Chengdu Baiyu Pharmaceutical
- Class Antineoplastics; Small molecules
- Mechanism of Action DNA-activated protein kinase inhibitors
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Orphan Drug Status
No
Orphan designation is assigned by a regulatory body to encourage companies to develop drugs for rare diseases.
- New Molecular Entity Yes
Highest Development Phases
- Phase I/II Prostate cancer; Solid tumours
Most Recent Events
- 16 Dec 2025 Phase-I/II clinical trials in Prostate cancer (Combination therapy, Hormone refractory, Metastatic disease, Second-line therapy or greater) in Australia (unspecified route) (NCT07226986)
- 12 Nov 2025 Novartis Pharmaceuticals plans a phase Ib/II trial for Prostate cancer (Combination therapy, Hormone refractory, Metastatic disease, Second-line therapy or greater) in December 2025 (PO) (NCT07226986)
- 18 Oct 2024 Chengdu Baiyu Pharmaceutical terminates a phase Ib/II trial in Solid tumours (Late-stage disease, Second-line therapy or greater) in China due to the sponsor adjusts the clinical development strategy (PO) (NCT06524804)