XS 03
Alternative Names: XS-03Latest Information Update: 04 Jul 2025
At a glance
- Originator XSXH Therapeutics
- Class Antineoplastics; Small molecules
- Mechanism of Action Polo-like kinase 1 inhibitors
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Orphan Drug Status
Orphan designation is assigned by a regulatory body to encourage companies to develop drugs for rare diseases.
- New Molecular Entity Yes
Highest Development Phases
- Preclinical Colorectal cancer
Most Recent Events
- 20 Apr 2025 XSXH Therapeutics in collaboration with NovaOnco Therapeutics plans a phase I/II trial for Colorectal cancer (Combination therapy, Late-stage disease, Metastatic disease) in China (PO), in June 2025 (NCT06936527)
- 27 Feb 2025 Preclinical trials in Colorectal cancer in China (PO), prior to February 2025
- 27 Feb 2025 The National Medical Products Administration (NMPA) approves clinical trial application for XS 03 in Colorectal cancer (Combination therapy, Late-stage disease, Metastatic disease) in China