BG 75202
Alternative Names: BG-75202Latest Information Update: 02 Jan 2026
At a glance
- Originator BeOne Medicines
- Class Antineoplastics; Small molecules
- Mechanism of Action KAT6A protein inhibitors; KAT6B protein inhibitors
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Orphan Drug Status
No
Orphan designation is assigned by a regulatory body to encourage companies to develop drugs for rare diseases.
- New Molecular Entity Yes
Highest Development Phases
- Phase I Breast cancer; Solid tumours
Most Recent Events
- 11 Dec 2025 Phase-I clinical trials in Breast cancer (Combination therapy, Late-stage disease, Metastatic disease) in Australia (PO) (NCT07222267)
- 11 Dec 2025 Phase-I clinical trials in Breast cancer (Combination therapy, Late-stage disease, Metastatic disease) in USA (PO) (NCT07222267)
- 11 Dec 2025 Phase-I clinical trials in Breast cancer (Late-stage disease, Metastatic disease, Monotherapy) in USA (PO) (NCT07222267)