Lutetium 177 DOTA HYNIC panPSMA - Telix Pharmaceuticals
Alternative Names: 177Lu-DOTA-HYNIC-panPSMA; [177Lu]Lu-PSMA; Lutetium-177-DOTA-HYNIC-panPSMA - Telix Pharmaceuticals; TLX597 TxLatest Information Update: 11 May 2026
At a glance
- Originator Telix Pharmaceuticals
- Class Antineoplastics; Radioisotopes; Radiopharmaceuticals; Small molecules
- Mechanism of Action Ionising radiation emitters
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Orphan Drug Status
No
Orphan designation is assigned by a regulatory body to encourage companies to develop drugs for rare diseases.
- New Molecular Entity Yes
Highest Development Phases
- Phase II Prostate cancer
Most Recent Events
- 30 Apr 2026 Telix Pharmaceuticals plans a phase II OPTIMAL-E trial for Prostate cancer (mHSPC)
- 07 Apr 2026 Pharmacokinetics data from a preclinical studies in Prostate cancer released by Telix Pharmaceuticals
- 16 Jun 2025 Phase-II clinical trials in Prostate cancer (Hormone refractory, Metastatic disease, Second line therapy or greater) in Australia (IV) (ACTRN12625000971437)