A Phase 1b, Open Label, 2-Part Study to Evaluate the Effect of Pelabresib (DAK539/CPI-0610) on the Pharmacokinetics of Repaglinide, Midazolam, and Combined Drospirenone/Ethinyl Estradiol Oral Contraceptive in Patients With Advanced Malignancies
Latest Information Update: 22 Jan 2026
At a glance
- Drugs Pelabresib (Primary) ; Drospirenone; Ethinylestradiol; Midazolam; Repaglinide
- Indications Cancer
- Focus Pharmacokinetics
- Sponsors Novartis Pharmaceuticals
Most Recent Events
- 22 Jan 2026 New trial record